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Artemether CAS 71963-77-4 Artemisia Annua Extract

Artemether CAS 71963-77-4 Fitar da Hoton Artemisia Annua

Cikakken Bayani

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Bambancin Sinadaran N/A
Cas No 71963-77-4
Tsarin sinadarai Saukewa: C16H26O5
Nauyin kwayoyin halitta 298.37
EINECS no. 663-549-0
Wurin narkewa 86-88 ° C
Wurin tafasa 359.79 ° C (ƙananan ƙididdiga)
Takamaiman juyawa D19.5+171°(c=2.59inCHCl3)
Yawan yawa 1.0733
Index na refraction 1.6200 (kimantawa)
Yanayin ajiya Yanayin ɗaki
Solubility DMSO≥20mg/ml
Bayyanar Foda
Makamantu Artemetherum/Artemtherin/Dihydroartemisininmethylether
Solubility Mai narkewa a cikin Ruwa
Categories Cire Shuka, Kari, Kula da Lafiya
Aikace-aikace Maganin zazzabin cizon sauro

Artemether shine lactone sesquiterpene wanda aka samo a cikin tushenArtemisia shekara, wanda aka fi sani da tsutsa mai dadi.Maganin maganin zazzabin cizon sauro ne mai ƙarfi wanda ake amfani da shi don magance da kuma hana cizon sauro.An fara fitar da Artemisinin, wanda ya kasance farkon fasahar artemether, daga shukar a shekarun 1970, kuma bincikensa ya sa wani mai bincike na kasar Sin Tu Youyou ya samu lambar yabo ta Nobel a fannin likitanci a shekarar 2015.

Artemether yana aiki ta hanyar lalata ƙwayoyin cuta da ke haifar da cutar zazzabin cizon sauro.Cutar zazzabin cizon sauro na faruwa ne ta hanyar wata kwayar cuta mai suna Plasmodium, wacce ke kamuwa da ita ga mutane ta hanyar cizon sauro na Anopheles mata masu dauke da cutar.Da zarar sun shiga cikin mahallin ɗan adam, ƙwayoyin cuta suna ƙaruwa da sauri a cikin hanta da jajayen ƙwayoyin jini, suna haifar da zazzaɓi, sanyi, da sauran alamun mura.Idan ba a kula da shi ba, zazzabin cizon sauro na iya yin kisa.

Artemether yana da matukar tasiri a kan nau'ikan Plasmodium falciparum masu jure magunguna, wanda ke haifar da mafi yawan mace-mace masu nasaba da zazzabin cizon sauro a duniya.Hakanan yana da tasiri akan sauran nau'ikan ƙwayoyin cuta na Plasmodium waɗanda ke haifar da zazzabin cizon sauro.Artemether yawanci ana gudanar da shi tare da wasu magunguna, kamar lumefantrine, don rage haɗarin juriya na ƙwayoyi.

Baya ga amfani da shi azaman maganin zazzabin cizon sauro, an kuma gano artemether yana da sauran abubuwan warkewa.Nazarin ya nuna cewa yana da maganin kumburi, anti-tumor, da kuma maganin cutar hoto.An yi amfani da shi don magance cututtukan arthritis, lupus, da sauran cututtuka na autoimmune.Hakanan an bincika don yuwuwar ta don kula da COVID-19, kodayake ana buƙatar ƙarin bincike don tabbatar da ingancin sa.

Artemether gabaɗaya yana da aminci kuma ana jurewa sosai lokacin amfani da shi kamar yadda aka umarce shi.Koyaya, kamar duk kwayoyi, yana iya haifar da illa.Mafi yawan illolin da ke tattare da artemether sun haɗa da tashin zuciya, amai, juwa, da ciwon kai.A lokuta da ba kasafai ba, yana iya haifar da munanan halayen halayen, kamar bugun zuciya, tashin hankali, da lalacewar hanta.

A ƙarshe, artemether magani ne mai ƙarfi na rigakafin zazzabin cizon sauro wanda ya canza maganin zazzabin cizon sauro da rigakafin.Bincikensa ya ceci rayuka marasa adadi kuma ya sami karɓuwa ga al'ummar kimiyya.Sauran kaddarorinsa na warkewa sun sa ya zama ɗan takara mai ban sha'awa don maganin wasu cututtuka.Ko da yake yana iya haifar da illa, amfanin sa ya zarce kasadarsa idan aka yi amfani da shi a ƙarƙashin kulawar likita.
Siffofin da aka saba amfani da su sun haɗa da allunan, capsules da allurai.Nau'o'in magungunan sune magungunan rigakafin zazzabin cizon sauro, kuma babban bangaren shine artemether.Halin sanadin allunan artemether shine farar allunan.Halin capsule na artemether shine capsule, abin da ke ciki shine farin foda;Halin miyagun ƙwayoyi na allurar artemether ba shi da launi zuwa haske mai launin rawaya - kamar ruwa.

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